Relative Selectivity of Covalent Inhibitors Requires Assessment of Inactivation Kinetics and Cellular Occupancy: A Case Study of Ibrutinib and Acalabrutinib

31st Annual Meeting and Associated Programs of the Society for Immunotherapy of Cancer (SITC 2016): part two

Pharmaceuticals, Free Full-Text

Relative Selectivity of Covalent Inhibitors Requires Assessment of Inactivation Kinetics and Cellular Occupancy: A Case Study of Ibrutinib and Acalabrutinib

Pharmaceuticals, Free Full-Text

Advances in covalent drug discovery

Case Study - COVALfinder to Study Irreversible EGFR Drugs

Kinetic mechanisms of covalent inhibition - ScienceDirect

31st Annual Meeting and Associated Programs of the Society for Immunotherapy of Cancer (SITC 2016): part two – topic of research paper in Biological sciences. Download scholarly article PDF and read for

Sulfamate Acetamides as Self-Immolative Electrophiles for Covalent Ligand-Directed Release Chemistry